Publications
Accelerating biomedical discoveries in brain health through transformative neuropathology of aging and neurodegeneration
Neuron. 2025 Nov 19. Murray ME, Smith C, Menon V, ..., Vogel JW, Dugger BN, Phatnani H.
An improved model for prediction of de novo designed proteins with diverse geometries
bioRxiv. 2025 Jun 06. Orr B, Crilly SE, Akpinaroglu D, Zhu E, Keiser MJ, Kortemme T.
Learning precise segmentation of neurofibrillary tangles from rapid manual point annotations
bioRxiv. 2024 May 15. Ghandian S, Albarghouthi L, Nava K, ..., Jin LW, Dugger BN, Keiser MJ.
Toward a generalizable machine learning workflow for neurodegenerative disease staging with focus on neurofibrillary tangles
Acta Neuropathol Commun. 2023 Dec 18. Vizcarra JC, Pearce TM, Dugger BN, ..., Glass JD, Farrell K, Gutman DA.
Autoregressive fragment-based diffusion for pocket-aware ligand design
arXiv - NeurIPS GenBio. 2023 Nov 2. Ghorbani M, Gendelev L, Beroza P, Keiser MJ.
A single-cell gene expression language model
arXiv - NeurIPS LMRL. 2022 Oct 25. Connell W, Khan U, Keiser MJ.
Stress testing reveals gaps in clinic readiness of image-based diagnostic artificial intelligence models
NPJ Digit Med. 2021 Jan 21. Young AT, Fernandez K, Pfau J, ..., Tam A, Keiser MJ, Wei ML.
Predicting Cellular Drug Sensitivity using Conditional Modulation of Gene Expression
bioRxiv - NeurIPS LMRL. 2020 Dec 11. Connell W, Keiser MJ.
Attention-Based Learning on Molecular Ensembles
arXiv - NeurIPS ML4Molecules. 2020 Nov 25. Chuang KV, Keiser MJ.
Learning Molecular Representations for Medicinal Chemistry
J Med Chem. 2020 Aug 27. Chuang KV, Gunsalus LM, Keiser MJ.
Artificial Intelligence in Dermatology: A Primer
J Invest Dermatol. 2020 Aug. Young AT, Xiong M, Pfau J, Keiser MJ, Wei ML.
Robust Semantic Interpretability: Revisiting Concept Activation Vectors
arXiv - ICML - WHI. 2020 Jul 17. Pfau J, Young AT, Wei J, Wei ML, Keiser MJ.
Global Saliency: Aggregating Saliency Maps to Assess Dataset Artefact Bias
arXiv - NeurIPS ML4H. 2019 Oct 16. Pfau J, Young AT, Wei ML, Keiser MJ.
Comment on "Predicting reaction performance in C-N cross-coupling using machine learning"
Science. 2018 Nov 16. Chuang KV, Keiser MJ.
Adversarial Controls for Scientific Machine Learning
ACS Chem Biol. 2018 Oct 19. Chuang KV, Keiser MJ.
Predicted Biological Activity of Purchasable Chemical Space
J Chem Inf Model. 2018 Jan 22. Irwin JJ, Gaskins G, Sterling T, Mysinger MM, Keiser MJ.
Zebrafish behavioral profiling identifies multitarget antipsychotic-like compounds
Nat Chem Biol. 2016 Jul. Bruni G, Rennekamp AJ, Velenich A, ..., Keiser MJ, Peterson RT, Kokel D.
Leveraging Large-scale Behavioral Profiling in Zebrafish to Explore Neuroactive Polypharmacology
ACS Chem Biol. 2016 Apr 15. McCarroll MN, Gendelev L, Keiser MJ, Kokel D.
Polygenic overlap between schizophrenia risk and antipsychotic response: a genomic medicine approach
Lancet Psychiatry. 2016 Apr. Ruderfer DM, Charney AW, Readhead B, ..., Purcell SM, Dudley JT, Sklar P.
Prediction and validation of enzyme and transporter off-targets for metformin
J Pharmacokinet Pharmacodyn. 2015 Oct. Yee SW, Lin L, Merski M, Keiser MJ, Gupta A, Zhang Y, Chien HC, Shoichet BK, Giacomini KM.
Systems pharmacology augments drug safety surveillance
Clin Pharmacol Ther. 2015 Feb. Lorberbaum T, Nasir M, Keiser MJ, Vilar S, Hripcsak G, Tatonetti NP.
In silico molecular comparisons of C. elegans and mammalian pharmacology identify distinct targets that regulate feeding
PLoS Biol. 2013 Nov. Lemieux GA, Keiser MJ, Sassano MF, Laggner C, Mayer F, Bainton RJ, Werb Z, Roth BL, Shoichet BK, Ashrafi K.
Large-scale prediction and testing of drug activity on side-effect targets
Nature. 2012 Jun 10. Lounkine E, Keiser MJ, Whitebread S, ..., Cote S, Shoichet BK, Urban L.
Chemical informatics and target identification in a zebrafish phenotypic screen
Nat Chem Biol. 2011 Dec 18. Laggner C, Kokel D, Setola V, ..., Roth BL, Peterson RT, Shoichet BK.
The presynaptic component of the serotonergic system is required for clozapine's efficacy
Neuropsychopharmacology. 2011 Feb. Yadav PN, Abbas AI, Farrell MS, ..., Gingrich J, Beck SG, Roth BL.
Complementarity between a docking and a high-throughput screen in discovering new cruzain inhibitors
J Med Chem. 2010 Jul 8. Ferreira RS, Simeonov A, Jadhav A, Eidam O, Mott BT, Keiser MJ, McKerrow JH, Maloney DJ, Irwin JJ, Shoichet BK.
Prediction and evaluation of protein farnesyltransferase inhibition by commercial drugs
J Med Chem. 2010 Mar 25. DeGraw AJ, Keiser MJ, Ochocki JD, Shoichet BK, Distefano MD.
A pilot study of the pharmacodynamic impact of SSRI drug selection and beta-1 receptor genotype (ADRB1) on cardiac vital signs in depressed patients: a novel pharmacogenetic approach
Psychopharmacol Bull. 2010. Thomas KL, Ellingrod VL, Bishop JR, Keiser MJ.
Predicting new molecular targets for known drugs
Nature. 2009 Nov 12. Keiser MJ, Setola V, Irwin JJ, ..., Edwards DD, Shoichet BK, Roth BL.
A mapping of drug space from the viewpoint of small molecule metabolism
PLoS Comput Biol. 2009 Aug. Adams JC, Keiser MJ, Basuino L, Chambers HF, Lee DS, Wiest OG, Babbitt PC.
Quantifying biogenic bias in screening libraries
Nat Chem Biol. 2009 Jul. Hert J, Irwin JJ, Laggner C, Keiser MJ, Shoichet BK.
Off-target networks derived from ligand set similarity
Methods Mol Biol. 2009. Keiser MJ, Hert J.
Quantifying the relationships among drug classes
J Chem Inf Model. 2008 Apr. Hert J, Keiser MJ, Irwin JJ, Oprea TI, Shoichet BK.
Relating protein pharmacology by ligand chemistry
Nat Biotechnol. 2007 Feb. Keiser MJ, Roth BL, Armbruster BN, Ernsberger P, Irwin JJ, Shoichet BK.